6PXX
Class D beta-lactamase in complex with beta-lactam antibiotic
Summary for 6PXX
Entry DOI | 10.2210/pdb6pxx/pdb |
Descriptor | Beta-lactamase, (2~{S},3~{R})-3-methyl-2-[(2~{S},3~{R})-3-oxidanyl-1-oxidanylidene-butan-2-yl]-4-[(3~{S},5~{S})-5-[(sulfamoylamino)methyl]pyrrolidin-3-yl]sulfanyl-3,4-dihydro-2~{H}-pyrrole-5-carboxylic acid, 1,2-ETHANEDIOL, ... (6 entities in total) |
Functional Keywords | inhibitor, lactamase, hydrolase, hydrolase-antibiotic-inhibitor complex, hydrolase/antibiotic/inhibitor |
Biological source | Klebsiella pneumoniae |
Total number of polymer chains | 2 |
Total formula weight | 62141.84 |
Authors | |
Primary citation | Papp-Wallace, K.M.,Kumar, V.,Zeiser, E.T.,Becka, S.A.,van den Akker, F. Structural Analysis of The OXA-48 Carbapenemase Bound to A "Poor" Carbapenem Substrate, Doripenem. Antibiotics, 8:-, 2019 Cited by PubMed: 31514291DOI: 10.3390/antibiotics8030145 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.5 Å) |
Structure validation
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