6PBF
ZINC9155420-bound TRPV5 in nanodiscs
Summary for 6PBF
Entry DOI | 10.2210/pdb6pbf/pdb |
EMDB information | 20291 20292 |
Descriptor | Transient receptor potential cation channel subfamily V member 5, (1S)-1-(4-oxo-5-phenyl-3,4-dihydrothieno[2,3-d]pyrimidin-2-yl)ethyl [(2S)-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-2-yl]acetate (2 entities in total) |
Functional Keywords | trpv5, trp channel, inhibitor, calcium channel, transport protein |
Biological source | Oryctolagus cuniculus (Rabbit) |
Total number of polymer chains | 4 |
Total formula weight | 333508.84 |
Authors | Hughes, T.E.T.,Rosario, J.S.D.,Kapoor, A.,Yazici, A.T.,Fluck, E.C.,Filizola, M.,Rohacs, T.,Moiseenkova-Bell, V.Y. (deposition date: 2019-06-13, release date: 2019-11-06, Last modification date: 2024-03-20) |
Primary citation | Hughes, T.E.,Del Rosario, J.S.,Kapoor, A.,Yazici, A.T.,Yudin, Y.,Fluck, E.C.,Filizola, M.,Rohacs, T.,Moiseenkova-Bell, V.Y. Structure-based characterization of novel TRPV5 inhibitors. Elife, 8:-, 2019 Cited by PubMed: 31647410DOI: 10.7554/eLife.49572 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (4.2 Å) |
Structure validation
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