6OC0
Crystal structure of human DHODH with OSU-03012
Summary for 6OC0
Entry DOI | 10.2210/pdb6oc0/pdb |
Descriptor | Dihydroorotate dehydrogenase (quinone), mitochondrial, OROTIC ACID, FLAVIN MONONUCLEOTIDE, ... (6 entities in total) |
Functional Keywords | dhodh, inhibitor, osu-03012, oxidoreductase, oxidoreductase-oxidoreductase inhibitor complex, oxidoreductase/oxidoreductase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 41486.96 |
Authors | Durst, M.A.,Lavie, A. (deposition date: 2019-03-21, release date: 2019-11-13, Last modification date: 2023-10-11) |
Primary citation | Abt, E.R.,Rosser, E.W.,Durst, M.A.,Lok, V.,Poddar, S.,Le, T.M.,Cho, A.,Kim, W.,Wei, L.,Song, J.,Capri, J.R.,Xu, S.,Wu, N.,Slavik, R.,Jung, M.E.,Damoiseaux, R.,Czernin, J.,Donahue, T.R.,Lavie, A.,Radu, C.G. Metabolic Modifier Screen Reveals Secondary Targets of Protein Kinase Inhibitors within Nucleotide Metabolism. Cell Chem Biol, 27:197-, 2020 Cited by PubMed: 31734178DOI: 10.1016/j.chembiol.2019.10.012 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.4 Å) |
Structure validation
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