6LIM

BRD4-BD1 bound with compound 40

Summary for 6LIM

• Entry DOI: 10.2210/pdb6lim/pdb
• Descriptor: Bromodomain-containing protein 4, (3~{R})-6-[(4-isoquinolin-4-ylpyrimidin-2-yl)amino]-1,3-dimethyl-4-propan-2-yl-3~{H}-quinoxalin-2-one (3 entities in total)
• Functional Keywords: bromodomain, histone, gene regulation
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 1
• Total formula weight: 15192.60

Authors

Xiong, B.,Cao, D.,Li, Y. (deposition date: 2019-12-12, release date: 2020-12-16, Last modification date: 2023-11-22)

• Primary citation: Xiong, B.,Cao, D.; BRD4-BD1 bound with compound 40; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.75909502055 Å)