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6JYQ

Crystal structure of uPA_H99Y in complex with 3-azanyl-5-(azepan-1-yl)-N-carbamimidoyl-6-(furan-2-yl)pyrazine-2-carboxamide

Summary for 6JYQ
Entry DOI10.2210/pdb6jyq/pdb
DescriptorUrokinase-type plasminogen activator, 3-azanyl-5-(azepan-1-yl)-N-carbamimidoyl-6-(furan-2-yl)pyrazine-2-carboxamide, SULFATE ION, ... (4 entities in total)
Functional Keywordsurokinase, amiloride, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight28180.07
Authors
Buckley, B.,Jiang, L.G.,Huang, M.D.,Kelso, M.,Ranson, M. (deposition date: 2019-04-27, release date: 2020-05-13, Last modification date: 2024-10-16)
Primary citationBuckley, B.,Jiang, L.G.,Huang, M.D.,Kelso, M.,Ranson, M.
H99Y-6F-HMA-pH7
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.75 Å)
Structure validation

250059

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