6IIK
USP14 catalytic domain with IU1
Summary for 6IIK
Entry DOI | 10.2210/pdb6iik/pdb |
Descriptor | Ubiquitin carboxyl-terminal hydrolase 14, 1-[1-(4-fluorophenyl)-2,5-dimethyl-1H-pyrrol-3-yl]-2-(pyrrolidin-1-yl)ethan-1-one (3 entities in total) |
Functional Keywords | usp14 inhibitor complex, structural protein, hydrolase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 91810.27 |
Authors | Mei, Z.Q.,Wang, Y.W.,He, W.,Wang, F. (deposition date: 2018-10-06, release date: 2018-12-12, Last modification date: 2023-11-22) |
Primary citation | Wang, Y.,Jiang, Y.,Ding, S.,Li, J.,Song, N.,Ren, Y.,Hong, D.,Wu, C.,Li, B.,Wang, F.,He, W.,Wang, J.,Mei, Z. Small molecule inhibitors reveal allosteric regulation of USP14 via steric blockade. Cell Res., 28:1186-1194, 2018 Cited by PubMed: 30254335DOI: 10.1038/s41422-018-0091-x PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.97 Å) |
Structure validation
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