6HX8
Tubulin-STX3451 complex
Summary for 6HX8
Entry DOI | 10.2210/pdb6hx8/pdb |
Descriptor | Tubulin alpha-1B chain, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, PHOSPHOMETHYLPHOSPHONIC ACID ADENYLATE ESTER, ... (12 entities in total) |
Functional Keywords | cell cycle, tubulin fold, cytoskeleton, microtubule |
Biological source | Rattus norvegicus (Norway rat) More |
Total number of polymer chains | 6 |
Total formula weight | 265440.94 |
Authors | Dohle, W.,Prota, A.E.,Menchon, G.,Hamel, E.,Steinmetz, M.O.,Potter, B.V.L. (deposition date: 2018-10-16, release date: 2019-02-27, Last modification date: 2024-01-24) |
Primary citation | Dohle, W.,Prota, A.E.,Menchon, G.,Hamel, E.,Steinmetz, M.O.,Potter, B.V.L. Tetrahydroisoquinoline Sulfamates as Potent Microtubule Disruptors: Synthesis, Antiproliferative and Antitubulin Activity of Dichlorobenzyl-Based Derivatives, and a Tubulin Cocrystal Structure. ACS Omega, 4:755-764, 2019 Cited by PubMed: 30775645DOI: 10.1021/acsomega.8b02879 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.402 Å) |
Structure validation
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