6GQ7
PI3Kg IN COMPLEX WITH INH
Summary for 6GQ7
Entry DOI | 10.2210/pdb6gq7/pdb |
Descriptor | Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform, 3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-one (3 entities in total) |
Functional Keywords | pi3kg, inhibitor, complex, hydrolase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 111087.51 |
Authors | Petersen, J. (deposition date: 2018-06-07, release date: 2018-06-20, Last modification date: 2024-05-01) |
Primary citation | Petersen, J. PI3Kg IN COMPLEX WITH INH To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.84 Å) |
Structure validation
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