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6GDC

Human Carbonic Anhydrase II in complex with Benzenesulfonamide

Summary for 6GDC
Entry DOI10.2210/pdb6gdc/pdb
DescriptorCarbonic anhydrase 2, ZINC ION, MERCURY (II) ION, ... (8 entities in total)
Functional Keywordslyase, inhibitor, complex, co2-conversion
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight31068.98
Authors
Gloeckner, S.,Heine, A.,Klebe, G. (deposition date: 2018-04-23, release date: 2019-05-01, Last modification date: 2024-01-17)
Primary citationGlockner, S.,Ngo, K.,Sager, C.P.,Hufner-Wulsdorf, T.,Heine, A.,Klebe, G.
Conformational Changes in Alkyl Chains Determine the Thermodynamic and Kinetic Binding Profiles of Carbonic Anhydrase Inhibitors.
Acs Chem.Biol., 15:675-685, 2020
Cited by
PubMed: 32027480
DOI: 10.1021/acschembio.9b00895
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.079 Å)
Structure validation

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