6FQK
GluA2(flop) S729C ligand binding core dimer bound to ZK200775 at 1.98 Angstrom resolution
Summary for 6FQK
Entry DOI | 10.2210/pdb6fqk/pdb |
Descriptor | Glutamate receptor 2,Glutamate receptor 2, {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid (3 entities in total) |
Functional Keywords | ampar receptor, ligand binding domain, competitive antagonist, cross-linked dimer, membrane protein |
Biological source | Rattus norvegicus (Norway Rat) More |
Total number of polymer chains | 2 |
Total formula weight | 61652.41 |
Authors | Coombs, I.D.,Soto, D.,Gold, M.G.,Farrant, M.F.,Cull-Candy, S.G. (deposition date: 2018-02-14, release date: 2019-03-13, Last modification date: 2019-10-02) |
Primary citation | Coombs, I.D.,Soto, D.,McGee, T.P.,Gold, M.G.,Farrant, M.,Cull-Candy, S.G. Homomeric GluA2(R) AMPA receptors can conduct when desensitized. Nat Commun, 10:4312-4312, 2019 Cited by PubMed: 31541113DOI: 10.1038/s41467-019-12280-9 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.98010442598 Å) |
Structure validation
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