6FO6
CryoEM structure of bovine cytochrome bc1 in complex with the anti-malarial inhibitor SCR0911
Summary for 6FO6
Entry DOI | 10.2210/pdb6fo6/pdb |
EMDB information | 4286 4288 4292 |
Descriptor | Cytochrome b-c1 complex subunit Rieske, mitochondrial, PROTOPORPHYRIN IX CONTAINING FE, 7-methoxy-3-methyl-2-[5-[4-(trifluoromethyloxy)phenyl]pyridin-3-yl]quinolin-4-ol, ... (12 entities in total) |
Functional Keywords | cryo-em, inhibitor binding, membrane protein, cytochrome bc1 |
Biological source | Bos taurus (Bovine) More |
Total number of polymer chains | 18 |
Total formula weight | 504353.27 |
Authors | Johnson, R.M.,Amporndanai, K.,O'Neill, P.M.,Fishwick, C.W.G.,Jamson, A.H.,Rawson, S.D.,Hasnain, S.S.,Antonyuk, S.V.,Muench, S.P. (deposition date: 2018-02-06, release date: 2018-02-28, Last modification date: 2019-12-11) |
Primary citation | Amporndanai, K.,Johnson, R.M.,O'Neill, P.M.,Fishwick, C.W.G.,Jamson, A.H.,Rawson, S.,Muench, S.P.,Hasnain, S.S.,Antonyuk, S.V. X-ray and cryo-EM structures of inhibitor-bound cytochromebc1complexes for structure-based drug discovery. IUCrJ, 5:200-210, 2018 Cited by PubMed: 29765610DOI: 10.1107/S2052252518001616 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (4.1 Å) |
Structure validation
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