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6ELR

Human jak1 kinase domain in complex with compound 7

Summary for 6ELR
Entry DOI10.2210/pdb6elr/pdb
DescriptorTyrosine-Protein Kinase JAK1, [3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanol, SODIUM ION, ... (4 entities in total)
Functional Keywordsjanus kinase 1 kinase domain (jak1), transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight70367.27
Authors
Read, J.A. (deposition date: 2017-09-29, release date: 2018-10-10, Last modification date: 2024-11-13)
Primary citationgrimster, N.P.,read, J.A.
Human jak1 kinase domain in complex with compound 7
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.8 Å)
Structure validation

237423

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