6CPM
Structure of the USP15 deubiquitinase domain in complex with a third-generation inhibitory Ubv
Summary for 6CPM
Entry DOI | 10.2210/pdb6cpm/pdb |
Related | 6CRN 6CSI |
Descriptor | Ubiquitin carboxyl-terminal hydrolase 15, Ubiquitin variant 15.1d, CALCIUM ION, ... (8 entities in total) |
Functional Keywords | deubiuqitination, ubv, high-affinity, inhibition, signaling protein |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 4 |
Total formula weight | 99524.44 |
Authors | Singer, A.U.,Teyra, J.,Boehmelt, G.,Lenter, M.,Sicheri, F.,Sidhu, S.S. (deposition date: 2018-03-13, release date: 2019-01-23, Last modification date: 2024-04-03) |
Primary citation | Teyra, J.,Singer, A.U.,Schmitges, F.W.,Jaynes, P.,Kit Leng Lui, S.,Polyak, M.J.,Fodil, N.,Krieger, J.R.,Tong, J.,Schwerdtfeger, C.,Brasher, B.B.,Ceccarelli, D.F.J.,Moffat, J.,Sicheri, F.,Moran, M.F.,Gros, P.,Eichhorn, P.J.A.,Lenter, M.,Boehmelt, G.,Sidhu, S.S. Structural and Functional Characterization of Ubiquitin Variant Inhibitors of USP15. Structure, 27:590-, 2019 Cited by PubMed: 30713027DOI: 10.1016/j.str.2019.01.002 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.011 Å) |
Structure validation
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