6CNH
Human PRPF4B in complex with Rebastinib
Summary for 6CNH
Entry DOI | 10.2210/pdb6cnh/pdb |
Descriptor | Serine/threonine-protein kinase PRP4 homolog, 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1H-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-N-methylpyridine-2-carboxamide, SULFATE ION, ... (4 entities in total) |
Functional Keywords | kinase, inhibitor, dcc2036, structural genomics, structural genomics consortium, sgc, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 41821.23 |
Authors | Godoi, P.H.C.,Santiago, A.S.,Ramos, P.Z.,Fala, A.M.,Salmazo, A.P.T.,Counago, R.M.,Righetto, G.L.,Silva, P.N.B.,Gileadi, O.,Guimaraes, C.R.W.,Massirer, K.B.,Arruda, P.,Elkins, J.M.,Edwards, A.M.,Structural Genomics Consortium (SGC) (deposition date: 2018-03-08, release date: 2018-03-28, Last modification date: 2023-10-04) |
Primary citation | Godoi, P.H.C.,Santiago, A.S.,Ramos, P.Z.,Silva, P.N.B.,Righetto, G.L.,Guimaraes, C.R.W.,Massirer, K.B.,Arruda, P.,Elkins, J.M.,Edwards, A.M. Crystal structure of the human PRPF4B in complex with Rebastinib To be Published, |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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