6BQQ

Crystal Structure of the Human CAMKK2B in complex with BI2526

Summary for 6BQQ

• Entry DOI: 10.2210/pdb6bqq/pdb
• Descriptor: Calcium/calmodulin-dependent protein kinase kinase 2, 4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-N-(1-methylpiperidin-4-yl)benzamide, ACETATE ION, ... (4 entities in total)
• Functional Keywords: transferase, protein kinase domain, structural genomics, structural genomics consortium, sgc, transferase inhibitor complex
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 1
• Total formula weight: 33826.04

Authors

Counago, R.M.,de Souza, G.P.,dos Reis, C.V.,Ramos, P.Z.,Drewry, D.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC) (deposition date: 2017-11-28, release date: 2017-12-13, Last modification date: 2023-10-04)

• Primary citation: Counago, R.M.,de Souza, G.P.,dos Reis, C.V.,Drewry, D.,Massirer, K.B.,Arruda, P.,Edwards, A.M.,Elkins, J.M.,Structural Genomics Consortium (SGC); Crystal Structure of the Human CAMKK2B in complex with BI2526; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.8 Å)