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6B1L

Crystal structure of glycylpeptide N-tetradecanoyltransferase from Plasmodium vivax in complex with inhibitor IMP-0001173

Summary for 6B1L
Entry DOI10.2210/pdb6b1l/pdb
DescriptorGlycylpeptide N-tetradecanoyltransferase, TETRADECANOYL-COA, 1-(5-fluoro-2-{methyl[3-(methylamino)propyl]amino}pyrimidin-4-yl)-N-[(imidazo[1,2-a]pyridin-3-yl)methyl]azetidine-3-carboxamide, ... (4 entities in total)
Functional Keywordsssgcid, glycylpeptide n-tetradecanoyltransferase, n-myristoyltransferase, nmt, plasmodium vivax, salvador i, structural genomics, seattle structural genomics center for infectious disease, transferase
Biological sourcePlasmodium vivax (strain Salvador I)
Total number of polymer chains2
Total formula weight95906.27
Authors
Seattle Structural Genomics Center for Infectious Disease (SSGCID) (deposition date: 2017-09-18, release date: 2018-09-26, Last modification date: 2023-10-04)
Primary citationDranow, D.M.,Horanyi, P.S.,Lorimer, D.D.,Edwards, T.E.
Crystal structure of glycylpeptide N-tetradecanoyltransferase from Plasmodium vivax in complex with inhibitor IMP-0001173
to be published,
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

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