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6AG9

Crystal structure of uPA in complex with 3,5-bis(azanyl)-6-(1-benzofuran-2-yl)-N-carbamimidoyl-pyrazine-2- carboxamide

Summary for 6AG9
Entry DOI10.2210/pdb6ag9/pdb
DescriptorUrokinase-type plasminogen activator, 3,5-bis(azanyl)-6-(1-benzofuran-2-yl)-N-carbamimidoyl-pyrazine-2-carboxamide, SULFATE ION, ... (4 entities in total)
Functional Keywordsurokinase, amiloride, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight28849.73
Authors
Buckley, B.,Jiang, L.G.,Majed, H.,Huang, M.D.,Kelso, M.,Ranson, M. (deposition date: 2018-08-09, release date: 2019-09-18, Last modification date: 2023-11-22)
Primary citationBuckley, B.,Jiang, L.G.,Huang, M.D.,Kelso, M.,Ranson, M.
uPA-HMA
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.63 Å)
Structure validation

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