6A5X
FXR-LBD with HNC180 and SRC1
Summary for 6A5X
Entry DOI | 10.2210/pdb6a5x/pdb |
Related | 6A5W |
Descriptor | Bile acid receptor, Nuclear receptor coactivator 1, SULFATE ION, ... (5 entities in total) |
Functional Keywords | nuclear receptor, coactivator, agonist, complex, transcription |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 29336.20 |
Authors | |
Primary citation | Wang, N.,Zou, Q.,Xu, J.,Zhang, J.,Liu, J. Ligand binding and heterodimerization with retinoid X receptor alpha (RXR alpha ) induce farnesoid X receptor (FXR) conformational changes affecting coactivator binding J. Biol. Chem., 293:18180-18191, 2018 Cited by PubMed: 30275017DOI: 10.1074/jbc.RA118.004652 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
Download full validation report