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6YZ3

PqsR (MvfR) in complex with antagonist 19

This is a non-PDB format compatible entry.
Summary for 6YZ3
Entry DOI10.2210/pdb6yz3/pdb
Related6Z07 6Z17 6Z5K
DescriptorLysR family transcriptional regulator, 1,2-ETHANEDIOL, 6-chloranyl-3-[(2-hexyl-2,3-dihydro-1,3-thiazol-4-yl)methyl]quinazolin-4-one, ... (4 entities in total)
Functional Keywordspseudomonas aeruginosa, antagonist, quorum sensing, dna binding protein
Biological sourcePseudomonas aeruginosa
Total number of polymer chains1
Total formula weight27173.15
Authors
Richardson, W.K.,Emsley, J. (deposition date: 2020-05-06, release date: 2020-09-16, Last modification date: 2024-01-24)
Primary citationGrossman, S.,Soukarieh, F.,Richardson, W.,Liu, R.,Mashabi, A.,Emsley, J.,Williams, P.,Camara, M.,Stocks, M.J.
Novel quinazolinone inhibitors of the Pseudomonas aeruginosa quorum sensing transcriptional regulator PqsR.
Eur.J.Med.Chem., 208:112778-112778, 2020
Cited by
PubMed: 32927392
DOI: 10.1016/j.ejmech.2020.112778
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3 Å)
Structure validation

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