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6T0H

Crystal structure of CYP124 in complex with 1-alpha-hydroxy-vitamin D3

Summary for 6T0H
Entry DOI10.2210/pdb6t0h/pdb
DescriptorCYP124 in complex with inhibitor carbethoxyhexyl imidazole, PROTOPORPHYRIN IX CONTAINING FE, 1-alpha-hydroxy-vitamin D3, ... (8 entities in total)
Functional Keywordscytochrome, p450, cyp, oxidoreductase, 124, cyp124, vitamin, d3, vitamind3, 1 alpha-hydroxy, 1-alpha-hydroxy, alfacalcidol, calciferol, cholecalciferol, tuberculosis, mycobacterium tuberculosis
Biological sourceMycobacterium tuberculosis H37Rv
Total number of polymer chains1
Total formula weight51280.44
Authors
Bukhdruker, S.,Marin, E.,Varaksa, T.,Gilep, A.,Strushkevich, N.,Borshchevskiy, V. (deposition date: 2019-10-03, release date: 2020-10-14, Last modification date: 2024-02-07)
Primary citationVaraksa, T.,Bukhdruker, S.,Grabovec, I.,Marin, E.,Kavaleuski, A.,Gusach, A.,Kovalev, K.,Maslov, I.,Luginina, A.,Zabelskii, D.,Astashkin, R.,Shevtsov, M.,Smolskaya, S.,Kavaleuskaya, A.,Shabunya, P.,Baranovsky, A.,Dolgopalets, V.,Charnou, Y.,Savachka, A.,Litvinovskaya, R.,Hurski, A.,Shevchenko, E.,Rogachev, A.,Mishin, A.,Gordeliy, V.,Gabrielian, A.,Hurt, D.E.,Nikonenko, B.,Majorov, K.,Apt, A.,Rosenthal, A.,Gilep, A.,Borshchevskiy, V.,Strushkevich, N.
Metabolic Fate of Human Immunoactive Sterols in Mycobacterium tuberculosis.
J.Mol.Biol., 433:166763-166763, 2021
Cited by
PubMed: 33359098
DOI: 10.1016/j.jmb.2020.166763
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.18 Å)
Structure validation

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