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6RCH

Crystal structure of Casein kinase I isoform delta (CK1 delta) complexed with SR4133 inhibitor

Summary for 6RCH
Entry DOI10.2210/pdb6rch/pdb
DescriptorCasein kinase I isoform delta, SULFATE ION, 1,2-ETHANEDIOL, ... (6 entities in total)
Functional Keywordsck1 delta, ck1d, kinase inhibitor, structural genomics, structural genomics consortium, sgc, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight70452.95
Authors
Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2019-04-11, release date: 2020-03-25, Last modification date: 2024-01-24)
Primary citationChaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC)
Crystal structure of Casein kinase I isoform delta (CK1 delta) complexed with SR4133 inhibitor
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.45 Å)
Structure validation

246704

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