6RCG

Crystal structure of Casein kinase 1 delta (CK1 delta) complexed with SR3029 inhibitor

Summary for 6RCG

• Entry DOI: 10.2210/pdb6rcg/pdb
• Descriptor: Casein kinase I isoform delta, 1,2-ETHANEDIOL, ~{N}-[[6,7-bis(fluoranyl)-1~{H}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amine, ... (4 entities in total)
• Functional Keywords: csnk1d, ck1 delta, ck1d, kinase inhibitor, structural genomics, structural genomics consortium, sgc, transferase
• Biological source: Homo sapiens (Human)
• Total number of polymer chains: 1
• Total formula weight: 35029.39

Authors

Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC) (deposition date: 2019-04-11, release date: 2020-03-25, Last modification date: 2024-01-24)

• Primary citation: Chaikuad, A.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Roush, W.R.,Knapp, S.,Structural Genomics Consortium (SGC); Crystal structure of Casein kinase 1 delta (CK1 delta) complexed with SR3029 inhibitor; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.4 Å)