6QJU
Crystal structure of human Bromodomain containing protein 3 (BRD3) in complex with 3-bromo-1H-indazol-5-amine
Summary for 6QJU
Entry DOI | 10.2210/pdb6qju/pdb |
Descriptor | Bromodomain-containing protein 3, 1,2-ETHANEDIOL, THIOCYANATE ION, ... (7 entities in total) |
Functional Keywords | bromodomain, complex, inhibitor, ligand, halogen bonding, xb, heflib, halogen-enriched fragment library, signaling protein |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 2 |
Total formula weight | 29754.13 |
Authors | Braun, M.B.,Stehle, T.,Heidrich, J. (deposition date: 2019-01-25, release date: 2020-02-12, Last modification date: 2024-01-24) |
Primary citation | Braun, M.B.,Stehle, S.,Heidrich, J.,Boeckler, F.M. Br-O-modomain (BRD3) halogen binding to a small molecule To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.202 Å) |
Structure validation
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