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6QJU

Crystal structure of human Bromodomain containing protein 3 (BRD3) in complex with 3-bromo-1H-indazol-5-amine

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue EDO A 301
ChainResidue
AILE76
ATYR115
AHOH474
BTRP96

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 302
ChainResidue
ATRP57
AMET125
AHOH430
BTRP51

site_idAC3
Number of Residues4
Detailsbinding site for residue SCN A 303
ChainResidue
AASN92
ATYR94
AHOH413
ALYS88

site_idAC4
Number of Residues10
Detailsbinding site for residue J58 A 304
ChainResidue
APRO58
AVAL63
ATYR73
AASN111
ACYS112
ATYR115
AASN116
AHOH415
AHOH450
AHOH463

site_idAC5
Number of Residues6
Detailsbinding site for residue EDO B 300
ChainResidue
ALEU134
BILE76
BILE77
BLYS78
BASN79
BASN111

site_idAC6
Number of Residues3
Detailsbinding site for residue DMS B 301
ChainResidue
BVAL63
BASN116
BHOH411

site_idAC7
Number of Residues4
Detailsbinding site for residue NA B 302
ChainResidue
BTYR113
BILE114
BASN116
BHOH501

site_idAC8
Number of Residues5
Detailsbinding site for residue NA B 303
ChainResidue
BTHR36
BASN37
BGLN38
BGLU143
BHOH407

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFyqpvDaiklnlpDYHkiIknpMdmgtIkkrlenny..Ywsasecmqdfnt.MftNCyiY
ChainResidueDetails
AALA56-TYR115

221716

PDB entries from 2024-06-26

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