6JIO
Human LXR-beta in complex with a ligand
Summary for 6JIO
Entry DOI | 10.2210/pdb6jio/pdb |
Descriptor | Oxysterols receptor LXR-beta, tert-butyl 7-amino-3,4-dihydroisoquinoline-2(1H)-carboxylate (3 entities in total) |
Functional Keywords | nuclear receptor, dna binding protein |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 4 |
Total formula weight | 125182.99 |
Authors | |
Primary citation | Zhang, Z.,Chen, H.,Chen, Z.,Ding, P.,Ju, Y.,Gu, Q.,Xu, J.,Zhou, H. Identify liver X receptor beta modulator building blocks by developing a fluorescence polarization-based competition assay. Eur.J.Med.Chem., 178:458-467, 2019 Cited by PubMed: 31202993DOI: 10.1016/j.ejmech.2019.06.011 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
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