6BAB
The structure of human CamKII with bound inhibitor
Summary for 6BAB
Entry DOI | 10.2210/pdb6bab/pdb |
Descriptor | Calcium/calmodulin-dependent protein kinase type II subunit delta, N-[(2S)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide, L(+)-TARTARIC ACID, ... (4 entities in total) |
Functional Keywords | kinase, camkii, inhibitor, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Mus musculus (Mouse) |
Cellular location | Cell membrane, sarcolemma ; Peripheral membrane protein ; Cytoplasmic side : Q6PHZ2 |
Total number of polymer chains | 4 |
Total formula weight | 140311.10 |
Authors | |
Primary citation | Koltun, D.,Somoza, J.R. TBD To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.91 Å) |
Structure validation
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