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5XIH

Crystal Structure of Toxoplasma gondii Prolyl-tRNA Synthetase (TgPRS) in complex with inhibitor 5

Summary for 5XIH
Entry DOI10.2210/pdb5xih/pdb
Related5XIF 5XIG 5XII 5XIJ 5XIK 5XIL 5XIO 5XIP 5XIQ
DescriptorProlyl-tRNA synthetase (ProRS), PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, MAGNESIUM ION, ... (6 entities in total)
Functional Keywordsprotein translation, prs, synthetase, inhibitor, infectious disease, ligase
Biological sourceToxoplasma gondii (strain ATCC 50611 / Me49)
Total number of polymer chains4
Total formula weight235466.26
Authors
Jain, V.,Manickam, Y.,Sharma, A. (deposition date: 2017-04-26, release date: 2018-03-07, Last modification date: 2023-11-22)
Primary citationJain, V.,Yogavel, M.,Kikuchi, H.,Oshima, Y.,Hariguchi, N.,Matsumoto, M.,Goel, P.,Touquet, B.,Jumani, R.S.,Tacchini-Cottier, F.,Harlos, K.,Huston, C.D.,Hakimi, M.A.,Sharma, A.
Targeting Prolyl-tRNA Synthetase to Accelerate Drug Discovery against Malaria, Leishmaniasis, Toxoplasmosis, Cryptosporidiosis, and Coccidiosis
Structure, 25:1495-1505.e6, 2017
Cited by
PubMed: 28867614
DOI: 10.1016/j.str.2017.07.015
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.2 Å)
Structure validation

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