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5WXT

Crystal structure of uPA-S195A in complex with S2444

Summary for 5WXT
Entry DOI10.2210/pdb5wxt/pdb
Related5WXF 5WXO 5WXP 5WXQ 5WXR 5WXS
Related PRD IDPRD_002229
DescriptorUrokinase-type plasminogen activator chain B, (2R)-N-[2-[[(2S)-1-[[4-[bis(oxidanyl)amino]phenyl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-2-oxidanylidene-ethyl]-5-oxidanylidene-pyrrolidine-2-carboxamide (3 entities in total)
Functional Keywordsserine proteases, upa, pepetide inhibitors, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight28890.85
Authors
Jiang, L.,Huang, M. (deposition date: 2017-01-08, release date: 2018-07-11, Last modification date: 2023-11-22)
Primary citationJiang, L.,Huang, M.
Crystal structure of uPA-S195A in complex with S2444
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

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