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5WVD

Structure of Mnk1 in complex with DS12881479

Summary for 5WVD
Entry DOI10.2210/pdb5wvd/pdb
Related5WVJ 5WVL
DescriptorMAP kinase interacting serine/threonine kinase 1, SULFATE ION, 1-methyl-N-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamide (3 entities in total)
Functional Keywordskinase, kinase inhibitor, inactive conformation, transferase
Biological sourceHomo sapiens (Human)
Total number of polymer chains2
Total formula weight70189.81
Authors
Matsui, Y.,Hanzawa, H. (deposition date: 2016-12-24, release date: 2018-01-03, Last modification date: 2023-11-22)
Primary citationMatsui, Y.,Yasumatsu, I.,Yoshida, K.I.,Iimura, S.,Ikeno, Y.,Nawano, T.,Fukano, H.,Ubukata, O.,Hanzawa, H.,Tanzawa, F.,Isoyama, T.
A novel inhibitor stabilizes the inactive conformation of MAPK-interacting kinase 1.
Acta Crystallogr F Struct Biol Commun, 74:156-160, 2018
Cited by
PubMed: 29497019
DOI: 10.1107/S2053230X18002108
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3 Å)
Structure validation

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