5V7T
crystal structure of PARP14 bound to N-{4-[4-(diphenylmethoxy)piperidin-1-yl]butyl}[1,2,4]triazolo[4,3-b]pyridazin-6-amine inhibitor
Summary for 5V7T
Entry DOI | 10.2210/pdb5v7t/pdb |
Related | 5V7W |
Descriptor | Poly [ADP-ribose] polymerase 14, N-{4-[4-(diphenylmethoxy)piperidin-1-yl]butyl}[1,2,4]triazolo[4,3-b]pyridazin-6-amine (3 entities in total) |
Functional Keywords | human parp14, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus: Q460N5 |
Total number of polymer chains | 1 |
Total formula weight | 22558.08 |
Authors | |
Primary citation | Yoneyama-Hirozane, M.,Matsumoto, S.I.,Toyoda, Y.,Saikatendu, K.S.,Zama, Y.,Yonemori, K.,Oonishi, M.,Ishii, T.,Kawamoto, T. Identification of PARP14 inhibitors using novel methods for detecting auto-ribosylation. Biochem. Biophys. Res. Commun., 486:626-631, 2017 Cited by PubMed: 28315326DOI: 10.1016/j.bbrc.2017.03.052 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.3 Å) |
Structure validation
Download full validation report