5UXD
Crystal structure of macrolide 2'-phosphotransferase MphH from Brachybacterium faecium in complex with azithromycin
Summary for 5UXD
Entry DOI | 10.2210/pdb5uxd/pdb |
Related | 5UXA 5UXB 5UXC |
Descriptor | Macrolide 2'-phosphotransferase MphH, AZITHROMYCIN, SULFATE ION, ... (5 entities in total) |
Functional Keywords | antibiotic resistance, macrolide, cave bacterium, phosphotransferase, kinase, alpha/beta protein, azithromycin, structural genomics, center for structural genomics of infectious diseases, csgid, national institute of allergy and infectious diseases, niaid, transferase-antibiotic complex, transferase/antibiotic |
Biological source | Brachybacterium faecium (strain ATCC 43885 / DSM 4810 / NCIB 9860) |
Total number of polymer chains | 2 |
Total formula weight | 67078.09 |
Authors | Stogios, P.J.,Skarina, T.,Wawrzak, Z.,Yim, V.,Savchenko, A.,Anderson, W.F.,Center for Structural Genomics of Infectious Diseases (CSGID) (deposition date: 2017-02-22, release date: 2017-08-23, Last modification date: 2023-10-04) |
Primary citation | Pawlowski, A.C.,Stogios, P.J.,Koteva, K.,Skarina, T.,Evdokimova, E.,Savchenko, A.,Wright, G.D. The evolution of substrate discrimination in macrolide antibiotic resistance enzymes. Nat Commun, 9:112-112, 2018 Cited by PubMed: 29317655DOI: 10.1038/s41467-017-02680-0 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.7 Å) |
Structure validation
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