5UQ0

FGFR1 kinase domain complex with fragment 2,2-dimethyl-2,3-dihydrobenzofuran-7-carboxamide

Summary for 5UQ0

• Entry DOI: 10.2210/pdb5uq0/pdb
• Descriptor: Fibroblast growth factor receptor 1, 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide (3 entities in total)
• Functional Keywords: kinase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
• Biological source: Homo sapiens (Human)
• Cellular location: Cell membrane; Single-pass type I membrane protein: P11362
• Total number of polymer chains: 2
• Total formula weight: 71089.68

Authors

Paik, W.-K.,Squire, C.J. (deposition date: 2017-02-05, release date: 2017-02-22, Last modification date: 2023-10-04)

• Primary citation: Paik, W.-K.,Yosaatmadja, Y.,Leung, I.,Squire, C.J.; Fragment screening diverse active sites; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.3 Å)