5ULG
Crystal structure of RPE65 in complex with MB-008 and palmitate
Summary for 5ULG
Entry DOI | 10.2210/pdb5ulg/pdb |
Related | 5ul5 |
Descriptor | Retinoid isomerohydrolase, FE (II) ION, PALMITIC ACID, ... (7 entities in total) |
Functional Keywords | retinoid isomerase, non-heme iron enzyme, inhibitor, isomerase, isomerase-isomerase inhibitor complex, isomerase/isomerase inhibitor |
Biological source | Bos taurus (Bovine) |
Total number of polymer chains | 2 |
Total formula weight | 123702.14 |
Authors | Kiser, P.D.,Palczewski, K. (deposition date: 2017-01-24, release date: 2017-05-17, Last modification date: 2023-10-04) |
Primary citation | Kiser, P.D.,Zhang, J.,Badiee, M.,Kinoshita, J.,Peachey, N.S.,Tochtrop, G.P.,Palczewski, K. Rational Tuning of Visual Cycle Modulator Pharmacodynamics. J. Pharmacol. Exp. Ther., 362:131-145, 2017 Cited by PubMed: 28476927DOI: 10.1124/jpet.117.240721 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
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