5OWR

Human STK10 bound to dasatinib

Summary for 5OWR

• Entry DOI: 10.2210/pdb5owr/pdb
• Descriptor: Serine/threonine-protein kinase 10, N-(2-CHLORO-6-METHYLPHENYL)-2-({6-[4-(2-HYDROXYETHYL)PIPERAZIN-1-YL]-2-METHYLPYRIMIDIN-4-YL}AMINO)-1,3-THIAZOLE-5-CARBOXAMIDE, CALCIUM ION, ... (4 entities in total)
• Functional Keywords: kinase, structural genomics consortium, sgc, transferase
• Biological source: Homo sapiens (Human)
• Cellular location: Cell membrane ; Peripheral membrane protein : O94804
• Total number of polymer chains: 1
• Total formula weight: 34826.69

Authors

Szklarz, M.,Muniz, J.R.C.,Vollmar, M.,von Delft, F.,Bountra, C.,Knapp, S.,Edwards, A.M.,Arrowsmith, C.,Elkins, J.M. (deposition date: 2017-09-04, release date: 2017-09-13, Last modification date: 2024-05-01)

• Primary citation: Elkins, J.M.; Human STK10 bound to dasatinib; To Be Published,

Experimental method

X-RAY DIFFRACTION (2.3 Å)