5OUA
Crystal Structure of the Protein-Kinase A catalytic subunit from Criteculus Griseus in complex with compound RKp017
Summary for 5OUA
| Entry DOI | 10.2210/pdb5oua/pdb |
| Descriptor | cAMP-dependent protein kinase catalytic subunit alpha, cAMP dependent protein kinase inhibitor, beta-D-ribopyranose, ... (4 entities in total) |
| Functional Keywords | complex, peptidic ligand, transferase |
| Biological source | Cricetulus griseus (Chinese hamster) More |
| Total number of polymer chains | 2 |
| Total formula weight | 43317.05 |
| Authors | Mueller, J.M.,Heine, A.,Klebe, G. (deposition date: 2017-08-23, release date: 2018-09-05, Last modification date: 2020-07-29) |
| Primary citation | Mueller, J.M.,Kirschner, R.,Geyer, A.,Klebe, G. Conceptional Design of Self-Assembling Bisubstrate-like Inhibitors of Protein Kinase A Resulting in a Boronic Acid Glutamate Linkage Acs Omega, 2019 Cited by DOI: 10.1021/acsomega.8b02364PDB entries with the same primary citation |
| Experimental method | X-RAY DIFFRACTION (1.67 Å) |
Structure validation
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