5OKD
Crystal structure of bovine Cytochrome bc1 in complex with inhibitor SCR0911.
Summary for 5OKD
Entry DOI | 10.2210/pdb5okd/pdb |
Descriptor | Cytochrome b-c1 complex subunit 1, mitochondrial, Cytochrome b-c1 complex subunit 9, TETRAETHYLENE GLYCOL, ... (22 entities in total) |
Functional Keywords | electron transport, antimalarial inhibitor, qi site binder |
Biological source | Bos taurus (Bovine) More |
Cellular location | Mitochondrion inner membrane; Peripheral membrane protein; Matrix side: P31800 P23004 Mitochondrion inner membrane: P00130 P00129 P13271 P00126 Mitochondrion inner membrane ; Multi-pass membrane protein : P00157 Mitochondrion inner membrane; Single-pass membrane protein; Intermembrane side: P00125 Mitochondrion inner membrane ; Single-pass membrane protein : P13272 P13272 |
Total number of polymer chains | 10 |
Total formula weight | 259445.61 |
Authors | Amporndanai, K.,O'Neill, P.M.,Hasnain, S.S.,Antonyuk, S.V. (deposition date: 2017-07-25, release date: 2018-02-28, Last modification date: 2024-01-17) |
Primary citation | Amporndanai, K.,Johnson, R.M.,O'Neill, P.M.,Fishwick, C.W.G.,Jamson, A.H.,Rawson, S.,Muench, S.P.,Hasnain, S.S.,Antonyuk, S.V. X-ray and cryo-EM structures of inhibitor-bound cytochromebc1complexes for structure-based drug discovery. IUCrJ, 5:200-210, 2018 Cited by PubMed: 29765610DOI: 10.1107/S2052252518001616 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.1 Å) |
Structure validation
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