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5O7P

HER3 in complex with Fab MF3178

Summary for 5O7P
Entry DOI10.2210/pdb5o7p/pdb
DescriptorReceptor tyrosine-protein kinase erbB-3, MF3178 FAB light chain, MF3178 FAB heavy chain, ... (5 entities in total)
Functional Keywordsher3 ectodomain, complex, fab, immune system
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains3
Total formula weight124001.59
Authors
De Nardis, C.,Gros, P. (deposition date: 2017-06-09, release date: 2018-05-16, Last modification date: 2024-01-17)
Primary citationGeuijen, C.A.W.,De Nardis, C.,Maussang, D.,Rovers, E.,Gallenne, T.,Hendriks, L.J.A.,Visser, T.,Nijhuis, R.,Logtenberg, T.,de Kruif, J.,Gros, P.,Throsby, M.
Unbiased Combinatorial Screening Identifies a Bispecific IgG1 that Potently Inhibits HER3 Signaling via HER2-Guided Ligand Blockade.
Cancer Cell, 33:922-936.e10, 2018
Cited by
PubMed: 29763625
DOI: 10.1016/j.ccell.2018.04.003
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (4.5 Å)
Structure validation

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