5NXC
LIM Domain Kinase 1 (LIMK1) In Complex With PF-00477736
Summary for 5NXC
Entry DOI | 10.2210/pdb5nxc/pdb |
Descriptor | LIM domain kinase 1, (2~{R})-2-azanyl-2-cyclohexyl-~{N}-[2-(1-methylpyrazol-4-yl)-9-oxidanylidene-3,10,11-triazatricyclo[6.4.1.0^{4,13}]trideca-1,4,6,8(13),11-pentaen-6-yl]ethanamide (3 entities in total) |
Functional Keywords | kinase actin cytoskeleton inhibitor, transferase |
Biological source | Homo sapiens (Human) |
Cellular location | Cytoplasm: P53667 |
Total number of polymer chains | 1 |
Total formula weight | 36414.25 |
Authors | Mathea, S.,Salah, E.,Pike, A.C.W.,Bushell, S.,Carpenter, E.P.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Bullock, A.N.,Knapp, S. (deposition date: 2017-05-10, release date: 2017-05-24, Last modification date: 2024-01-17) |
Primary citation | Mathea, S.,Salah, E.,Pike, A.C.W.,Bushell, S.,Carpenter, E.P.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Bullock, A.N.,Knapp, S. LIM Domain Kinase (LIMK1) In Complex With PF-00477736 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.25 Å) |
Structure validation
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