5NIM
EthR complex
Summary for 5NIM
Entry DOI | 10.2210/pdb5nim/pdb |
Descriptor | HTH-type transcriptional regulator EthR, [1-(2-hydroxyethyl)pyrrolo[3,4-c]pyrazol-5-yl]-(5-propyl-1,2-oxazol-3-yl)methanone, SULFATE ION, ... (4 entities in total) |
Functional Keywords | tetr repressor, dna binding protein, protein ligand complex |
Biological source | Mycobacterium tuberculosis |
Total number of polymer chains | 1 |
Total formula weight | 24166.07 |
Authors | Pohl, E.,Tatum, N.J.,Cole, J.C.,Baulard, A.R. (deposition date: 2017-03-24, release date: 2017-11-15, Last modification date: 2017-12-27) |
Primary citation | Tatum, N.J.,Liebeschuetz, J.W.,Cole, J.C.,Frita, R.,Herledan, A.,Baulard, A.R.,Willand, N.,Pohl, E. New active leads for tuberculosis booster drugs by structure-based drug discovery. Org. Biomol. Chem., 15:10245-10255, 2017 Cited by PubMed: 29182187DOI: 10.1039/c7ob00910k PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.5 Å) |
Structure validation
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