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5LX3

CRYSTAL STRUCTURE OF VISFATIN IN COMPLEX WITH SAR154782.

Summary for 5LX3
Entry DOI10.2210/pdb5lx3/pdb
DescriptorNicotinamide phosphoribosyltransferase, 6-[4-[(6-azanylpyridin-3-yl)methylcarbamoylamino]-3-fluoranyl-phenyl]-2-(ethylamino)-~{N}-(2-piperidin-1-ylethyl)pyridine-3-carboxamide (3 entities in total)
Functional Keywordstransferase, nampt, inhibitor, drug design, cancer
Biological sourceHomo sapiens (Human)
Cellular locationNucleus : P43490
Total number of polymer chains2
Total formula weight112515.40
Authors
Bertrand, T.,Marquette, J.P. (deposition date: 2016-09-20, release date: 2017-10-25)
Primary citationBertrand, T.,Marquette, J.P.
CRYSTAL STRUCTURE OF VISFATIN IN COMPLEX WITH SAR154782.
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

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