5J5T
GLK co-crystal structure with aminopyrrolopyrimidine inhibitor
Summary for 5J5T
Entry DOI | 10.2210/pdb5j5t/pdb |
Descriptor | Mitogen-activated protein kinase kinase kinase kinase 3, 5-[2-(piperidin-4-yl)-1,3-thiazol-5-yl]-3-[(pyridin-4-yl)methoxy]pyridin-2-amine (3 entities in total) |
Functional Keywords | protein kinsae, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 42593.44 |
Authors | Silvian, L.F.,Marcotte, D. (deposition date: 2016-04-03, release date: 2016-10-26, Last modification date: 2024-04-03) |
Primary citation | Marcotte, D.,Rushe, M.,M Arduini, R.,Lukacs, C.,Atkins, K.,Sun, X.,Little, K.,Cullivan, M.,Paramasivam, M.,Patterson, T.A.,Hesson, T.,D McKee, T.,May-Dracka, T.L.,Xin, Z.,Bertolotti-Ciarlet, A.,Bhisetti, G.R.,Lyssikatos, J.P.,Silvian, L.F. Germinal-center kinase-like kinase co-crystal structure reveals a swapped activation loop and C-terminal extension. Protein Sci., 26:152-162, 2017 Cited by PubMed: 27727493DOI: 10.1002/pro.3062 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.85 Å) |
Structure validation
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