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5H3Q

Crystal Structure of TrkA kinase with ligand

Summary for 5H3Q
Entry DOI10.2210/pdb5h3q/pdb
DescriptorHigh affinity nerve growth factor receptor, 1-[(3S,4R)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)urea, 2,3-DIHYDROXY-1,4-DITHIOBUTANE, ... (5 entities in total)
Functional Keywordstrka inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight37325.97
Authors
Noritaka, F. (deposition date: 2016-10-26, release date: 2017-02-22, Last modification date: 2023-11-08)
Primary citationFuruya, N.,Momose, T.,Katsuno, K.,Fushimi, N.,Muranaka, H.,Handa, C.,Ozawa, T.,Kinoshita, T.
The juxtamembrane region of TrkA kinase is critical for inhibitor selectivity
Bioorg. Med. Chem. Lett., 27:1233-1236, 2017
Cited by
PubMed: 28159414
DOI: 10.1016/j.bmcl.2017.01.056
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.1 Å)
Structure validation

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