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5GID

Crystal structure of VDR in complex with DLAM-4 (C2 form)

Summary for 5GID
Entry DOI10.2210/pdb5gid/pdb
Related5GIC 5GIE
DescriptorVitamin D3 receptor, SRC1, (3R,5S)-5-[(2R)-2-[(1R,3aS,4E,7aR)-7a-methyl-4-[(2Z)-2-[(3S,5R)-2-methylidene-3,5-bis(oxidanyl)cyclohexylidene]ethylidene]-2,3,3a,5,6,7-hexahydro-1H-inden-1-yl]propyl]-3-methyl-3-oxidanyl-1-(4-phenylbutyl)pyrrolidin-2-one, ... (4 entities in total)
Functional Keywordsnuclear receptor, transcription
Biological sourceRattus norvegicus (Rat)
More
Total number of polymer chains2
Total formula weight29916.60
Authors
Asano, L.,Shimizu, T. (deposition date: 2016-06-23, release date: 2016-12-07, Last modification date: 2024-03-20)
Primary citationAsano, L.,Waku, T.,Abe, R.,Kuwabara, N.,Ito, I.,Yanagisawa, J.,Nagasawa, K.,Shimizu, T.
Regulation of the vitamin D receptor by vitamin D lactam derivatives.
Febs Lett., 590:3270-3279, 2016
Cited by
PubMed: 27500498
DOI: 10.1002/1873-3468.12348
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.151 Å)
Structure validation

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