5FFY
Crystal structure of the bromodomain of human BRPF1 in complex with a benzimidazole ligand
Summary for 5FFY
Entry DOI | 10.2210/pdb5ffy/pdb |
Descriptor | Peregrin, 4-ethyl-~{N}-(6-methoxy-1,3-dimethyl-2-oxidanylidene-benzimidazol-5-yl)benzenesulfonamide (3 entities in total) |
Functional Keywords | peregrin, moz-morf complex, transcription |
Biological source | Homo sapiens (Human) |
Cellular location | Nucleus : P55201 |
Total number of polymer chains | 1 |
Total formula weight | 14079.14 |
Authors | Tallant, C.,Savitsky, P.,Nunez-Alonso, G.,Kopec, J.,Fedorov, O.,Filippakopoulos, P.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Knapp, S. (deposition date: 2015-12-19, release date: 2015-12-30, Last modification date: 2024-01-10) |
Primary citation | Tallant, C.,Savitsky, P.,Nunez-Alonso, G.,Kopec, J.,Fedorov, O.,Filippakopoulos, P.,von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Knapp, S. Crystal structure of the bromodomain of human BRPF1 in complex with a benzimidazole ligand To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.55 Å) |
Structure validation
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