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5EZH

Structure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in complex with compound 21 at 1.7A resolution

Summary for 5EZH
Entry DOI10.2210/pdb5ezh/pdb
DescriptorHTH-type transcriptional regulator EthR, ~{N}-[(1-pyridin-2-ylpiperidin-4-yl)methyl]pyrrolidine-1-carboxamide, SULFATE ION, ... (4 entities in total)
Functional Keywordsethr, transcription, repressor, mycobacterium tuberculosis
Biological sourceMycobacterium tuberculosis
Total number of polymer chains1
Total formula weight25932.09
Authors
Surade, S.,Blaszczyk, M.,Nikiforov, P.O.,Abell, C.,Blundell, T.L. (deposition date: 2015-11-26, release date: 2016-02-03, Last modification date: 2024-01-10)
Primary citationNikiforov, P.O.,Surade, S.,Blaszczyk, M.,Delorme, V.,Brodin, P.,Baulard, A.R.,Blundell, T.L.,Abell, C.
A fragment merging approach towards the development of small molecule inhibitors of Mycobacterium tuberculosis EthR for use as ethionamide boosters.
Org.Biomol.Chem., 14:2318-2326, 2016
Cited by
PubMed: 26806381
DOI: 10.1039/c5ob02630j
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.7 Å)
Structure validation

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