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5EZH

Structure of Transcriptional Regulatory Repressor Protein - EthR from Mycobacterium Tuberculosis in complex with compound 21 at 1.7A resolution

Functional Information from GO Data
ChainGOidnamespacecontents
A0000976molecular_functiontranscription cis-regulatory region binding
A0003677molecular_functionDNA binding
A0003700molecular_functionDNA-binding transcription factor activity
A0005515molecular_functionprotein binding
A0005829cellular_componentcytosol
A0006355biological_processregulation of DNA-templated transcription
A0045892biological_processnegative regulation of DNA-templated transcription
A0046677biological_processresponse to antibiotic
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 841 A 301
ChainResidue
ALEU76
APHE184
APHE187
AHOH401
AHOH418
AVAL80
ATHR121
AGLY124
AGLN125
AVAL134
ALEU137
ATRP138
AGLU180

site_idAC2
Number of Residues9
Detailsbinding site for residue 841 A 302
ChainResidue
ALEU87
ATRP103
AGLY106
APHE110
AMET142
ATYR148
AASN176
AASN179
ATRP207

site_idAC3
Number of Residues2
Detailsbinding site for residue SO4 A 303
ChainResidue
AASP98
AARG99

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues60
DetailsDomain: {"description":"HTH tetR-type","evidences":[{"source":"PROSITE-ProRule","id":"PRU00335","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues19
DetailsDNA binding: {"description":"H-T-H motif","evidences":[{"source":"PROSITE-ProRule","id":"PRU00335","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsSite: {"description":"Inhibitor-binding"}
ChainResidueDetails

239492

PDB entries from 2025-07-30

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