5EPM
Ceratotoxin variant in complex with specific antibody Fab fragment
Summary for 5EPM
Entry DOI | 10.2210/pdb5epm/pdb |
Descriptor | Antibody Fab fragment heavy chain, Antibody Fab fragment light chain, Beta-theraphotoxin-Cm1a, ... (4 entities in total) |
Functional Keywords | ceratotoxin, random mutagenesis, nav1.7 ion chanel, toxin-immune system complex, toxin/immune system |
Biological source | Mus musculus More |
Cellular location | Secreted : P84507 |
Total number of polymer chains | 6 |
Total formula weight | 103716.28 |
Authors | Strop, P.,Shcherbatko, A.,Rossi, A. (deposition date: 2015-11-11, release date: 2016-05-04, Last modification date: 2023-09-27) |
Primary citation | Shcherbatko, A.,Rossi, A.,Foletti, D.,Zhu, G.,Bogin, O.,Galindo Casas, M.,Rickert, M.,Hasa-Moreno, A.,Bartsevich, V.,Crameri, A.,Steiner, A.R.,Henningsen, R.,Gill, A.,Pons, J.,Shelton, D.L.,Rajpal, A.,Strop, P. Engineering Highly Potent and Selective Microproteins against Nav1.7 Sodium Channel for Treatment of Pain. J.Biol.Chem., 291:13974-13986, 2016 Cited by PubMed: 27129258DOI: 10.1074/jbc.M116.725978 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.75 Å) |
Structure validation
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