5B8I
Crystal structure of Calcineurin A and Calcineurin B in complex with FKBP12 and FK506 from Coccidioides immitis RS
Summary for 5B8I
Entry DOI | 10.2210/pdb5b8i/pdb |
Descriptor | Serine/threonine-protein phosphatase, Calcineurin subunit B, variant, Peptidylprolyl isomerase, ... (10 entities in total) |
Functional Keywords | ssgcid, nih, niaid, sbri, uw, beryllium, phosphatase, calcineurin, fkbp12, fk506, structural genomics, seattle structural genomics center for infectious disease, hydrolase |
Biological source | Coccidioides immitis (strain RS) (Valley fever fungus) More |
Total number of polymer chains | 3 |
Total formula weight | 81217.37 |
Authors | Seattle Structural Genomics Center for Infectious Disease (SSGCID),Fox III, D.,Dranow, D.M.,Lorimer, D.D.,Edwards, T.E. (deposition date: 2015-05-03, release date: 2015-05-20, Last modification date: 2023-09-27) |
Primary citation | Juvvadi, P.R.,Fox 3rd, D.,Bobay, B.G.,Hoy, M.J.,Gobeil, S.M.C.,Venters, R.A.,Chang, Z.,Lin, J.J.,Averette, A.F.,Cole, D.C.,Barrington, B.C.,Wheaton, J.D.,Ciofani, M.,Trzoss, M.,Li, X.,Lee, S.C.,Chen, Y.L.,Mutz, M.,Spicer, L.D.,Schumacher, M.A.,Heitman, J.,Steinbach, W.J. Harnessing calcineurin-FK506-FKBP12 crystal structures from invasive fungal pathogens to develop antifungal agents. Nat Commun, 10:4275-4275, 2019 Cited by PubMed: 31537789DOI: 10.1038/s41467-019-12199-1 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.85 Å) |
Structure validation
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