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5ALB

Ticagrelor antidote candidate MEDI2452 in complex with ticagrelor

Summary for 5ALB
Entry DOI10.2210/pdb5alb/pdb
Related5ALC
DescriptorMEDI2452 HEAVY CHAIN, MEDI2452 LIGHT CHAIN, Ticagrelor, ... (4 entities in total)
Functional Keywordsimmune system, antibody fragment, antidote, drug
Biological sourceHOMO SAPIENS (HUMAN)
More
Total number of polymer chains2
Total formula weight48014.33
Authors
Primary citationBuchanan, A.,Newton, P.,Pehrsson, S.,Inghardt, T.,Antonsson, T.,Svensson, P.,Sjogren, T.,Oster, L.,Janefeldt, A.,Sandinge, A.,Keyes, F.,Austin, M.,Spooner, J.,Gennemark, P.,Penney, M.,Howells, G.,Vaughan, T.,Nylander, S.
Structural and Functional Characterisation of a Specific Antidote for Ticagrelor.
Blood, 125:3484-, 2015
Cited by
PubMed: 25788700
DOI: 10.1182/BLOOD-2015-01-622928
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.16 Å)
Structure validation

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