5WXT
Crystal structure of uPA-S195A in complex with S2444
Summary for 5WXT
Entry DOI | 10.2210/pdb5wxt/pdb |
Related | 5WXF 5WXO 5WXP 5WXQ 5WXR 5WXS |
Related PRD ID | PRD_002229 |
Descriptor | Urokinase-type plasminogen activator chain B, (2R)-N-[2-[[(2S)-1-[[4-[bis(oxidanyl)amino]phenyl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-2-oxidanylidene-ethyl]-5-oxidanylidene-pyrrolidine-2-carboxamide (3 entities in total) |
Functional Keywords | serine proteases, upa, pepetide inhibitors, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 28890.85 |
Authors | |
Primary citation | Jiang, L.,Huang, M. Crystal structure of uPA-S195A in complex with S2444 To Be Published, |
Experimental method | X-RAY DIFFRACTION (2.1 Å) |
Structure validation
Download full validation report